I-Drotaverin i-anotpasmodic i-myotropic ine-action vasodilating. Isilwanyana sisincoko (isifananiselo esifanelekileyo) sesilwanyana esidumile njengeNo-shpa .
Ukubunjwa kunye nefomu yokukhululwa kweDottaverine
I-Drotaverine ifumaneka kwindlela yamacwecwe kunye nesisombululo sokujova.
Kwisinye ipilisi yesilwanyana iqulethe 40 mg ye drotaverine ngendlela ye-hydrochloride, kunye nezinto ezincedisayo-i-lactose, isitashi, i-povidone, i-magnesium stearate. Ukongezelela, kukho iipilisi zikaDottaverin, apho uxinzelelo lwezinto ezisebenzayo ngu-80 mg. Iibhilethi ziluphuzi, zincinci, i-biconvex, zipakishwe kwiibhanti ezili-10 kunye neepakethi zekhadibhodi. I-Drotaverine kwi-ampoules isetyenziselwa i-intramuscular (inqabile kakhulu-ye-intravenous). Elinye i-ampoule iqulethe i-2 ml yesisombululo kunye nokuxilongwa kwezinto ezixakekileyo ze-20 mg / ml.
Yintoni eyenza i-Drotaverine?
I-Drotaverin inciphisa ithoni kunye ne-motility ye-muscle epholileyo, iyibuyisela kwaye isuse i-spasms, iyanciphisa ngokukhawuleza imithanjeni yegazi, inemiphumo emihle ye-hypotensive.
I-Drotaverin isetyenziselwa ukufumana iintlungu ezahlukeneyo zendalo, nangona kungenjalo. Oku kubangelwa kukuba intlungu ayiyona isifo, kodwa isifo. Ngokususa i-spasm yeemisipha okanye imithana yegazi, i-drotaverin iyakususa isizathu esibangela intlungu. Yingakho i-Drotaverin isoloko isinceda ngeentloko kunye nentlungu yokuya esikhathini. Ngeentlungu ezibangelwa utyhafu, ukuvuvukala okanye ezinye iinkqubo zokugula, le nkunkuma ayinayo kwaye ayinayo impembelelo.
I-Drotaverine isetyenziswa:
- Ngama-spasms of muscle ephathekayo yezitho zangaphakathi (cholecystitis, cholangitis, cholecystolithiasis, cholangiolithiasis, papillitis, i-spastic colitis, intestinal colic).
- Ukunciphisa ama-spasms kwizifo ze-genitourinary system (nephrolithiasis, cystitis, pyelitis, ureterolithiasis, proctitis ).
- Ngezinye izifo zentsholongwane, kwindawo yokuqala - intlungu ngokuya esikhathini. Ukongezelela, isetyenziselwa ukuphelisa iintlobo zeengcambu ezihamba kakuhle zesisu ngexesha lokukhulelwa.
- Ngeentloko ezibangelwa ukuxinezeleka, ukungabikho kokulala, ukunyuka kwengqondo kwengqondo, ukhathazeka ngokomzimba (ikakhulukazi umxube wesifo kummandla wesibeleko). I-Drotaverine inokukunceda neentloko ezibangelwa ukunyuka kwengcinezelo yegazi, kodwa kule meko kusebenza ngokugqithisileyo kunye nokusetyenziswa kweziyobisi ezingekho komzimba.
- Njengesixhobo sokulungiselela ezinye iinkqubo zokuxilonga kunye nezonyango (i-catheterization of ureters, cholecystography).
- I-Drotaverine kunye ne-analgin yindlela eyaziwayo yokunciphisa izinga lokushisa, elidla ngokusebenza ngokuthe ngempumelelo kunezo-antipyretic ezikhethekileyo.
Ukungqinelana kokulawulwa kweDottaverine
Isilwayo siyaphikisana apha:
- i-hepatic, i-renal okanye i-heart failure;
- ukusilela i-lactose;
- i-adenoma yeprostate;
- glaucoma yokuvala i-angle.
Isetyenziswe ngokuqapha kwi-atherosclerosis yeerterotic coronary kunye nexinzelelo oluphantsi loxinzelelo.
Isistim nokuLawula
Iibhulethi zidakiwe kunanini na imini, ngaphandle kokuhlafuna. Thatha isiyobisi singaphaya kwama-80 mg (iipilisi ezi-2) ngexesha lokufumana, ukufika kathathu ngosuku. Isiphumo siqala ukuqala malunga nemizuzu eyi-15 emva kokulawula, kodwa ukuphumelela okuphezulu kufumaneka emva kwemizuzu engama-40-45.
I-Drotaverina injections yenziwe nge-intramuscularly, 1-2 ampoules (ukuya kuma-80 mg wezinto ezisetyenziswayo) nganye. Isiphumo sigqalwa 2 imizuzu emva kwejojo.
Isilwanyana senzelwe unyango olumqondiso, kwaye iintsuku ezingama-3 ngaphandle kokubonisana nodokotela ukuba asebenzise oko akucebisi.