I-Hypothiazide yiyilisi ephuma kwiqela le-thiazide diuretics . Iyeza linikezwa ngeefomethe. Ukuqhubela phambili siya kuqwalasela, sisiphi isicelo se-Hypothiazide kwiipilisi eziqeshwe okanye ezikhethiweyo, yintoni na ukuchasene kunye nemigangatho yokuhambisa.
Ukubunjwa kunye nesenzo se-pharmacological ye-Hypothiazide
Isithako esisebenzayo seHypothiazide yi-hydrochlorothiazide. Njengoko izinto ezincedisayo ekubunjweni kwamacwecwe zibandakanya ezo zithako:
- talc;
- gelatin;
- i-magnesium stearate;
- isitashi;
- lactose monohydrate.
I-Hypothiazide yi-diuretic leyo, ngaphezu koko, inefuthe elimelana ne-antihypertensive level in high blood pressure level. Umgaqo wempatho zokwelapha zamacwecwe uhambelana nomphumo wokuvimbela i-hydrochlorothiazide ekusebenzeni kwe-epithelium yamathambo e-renal. Oku kubonakaliswe, ngokukodwa, ekunciphiseni ukuchithwa kwe-sodium, i-chlorine (kunye nenani elincinci le-potassium kunye ne-bicarbonates) kunye namanani ahambelana namanzi. Kukho ukunciphisa ukuphuma kwe-iric acid kunye ne-calcium ions kunye nokwanda kwe-ion magnesium ions. I-Hypothiazide yeMithi inefuthe kwiimpawu ezahlukeneyo ze-asidi-base balance of body - zombini nge-acidification (acidosis) kunye ne-alkosis (alkalosis).
Ngokunciphisa umthamo we-extracellular fluid ephunyeziweyo ngokususa i-sodium, i-chlorine kunye ne-ion yamanzi, kunye nokwandisa imirhobho encinci, inyathelo elixhomekeke kuyo. Kule meko, isilwanyana asinasiphumo kwixinzelelo lwengcinezelo yegazi kwaye ayibangeli umphumo wokulutha. Isenzo se-hypotensive se-Hypothiazide sanda ngokutya okunesityu. Kwakhona, isichengisi sinceda ukunciphisa uxinzelelo lwe-intraocular.
Ngokusetyenziswa kwexesha elide, inkunkuma esebenzayo yeziyobisi inceda ukulibazisa ukuphuma kwee-calcium ngeentso, ezinokuthi zibe nefuthe elihle phambi kweentsimbi zeentso ezinee-calcium.
Iimpawu kunye nokuchasene nokusetyenziswa kwe-Hypothiazide
Iipilisi ze-Hypothiazidi zihlala zichazwe ngokuvuvukala kunye nokunyuka kwengcinezelo yegazi. Ngokwemiyalelo, uluhlu olupheleleyo lwezalathisi zezi ziza zilandelayo:
1. Iingongoma zengcinezelo ze-Arterial I kunye ne-II (njengendlela yokwenza i-monotherapy okanye ngokudibanisa nezinye iindlela zokwenza amanyathelo angama-antihypertensive action).
2. I-Edema yemvelaphi eyahlukileyo, ehambelana nayo:
- nephrotic syndrome;
- isifo sengqondo esingapheliyo okanye ukungaqiniseki kwamanzi;
- isifo soxinzelelo lwangaphambili;
- i-cirrhosis yesibindi;
- glomerulonephritis;
- ukufumana i-hormonal, njl njl.
3. Iimfuneko zokuthintela ukukhupha umchamo (ikakhulukazi kwi-nephrogenic insipidus).
4. Imfuno yokuthintela ukwakheka kwamatye kwiphepha le-urinary.
5. I- Glaucoma (kwinkqubo enzima).
Ukungqinelana kokuthatha i-Hypothiazide:
- anuria;
- utywala obunzima okanye ukungaqiniseki ngokuthe tye;
- isifo sikashukela sikwimeko eqinile;
- ukungaqiniseki kwamanqanaba;
- ukukhulelwa (i-trimester);
- i-hypokalemia engabonakaliyo, hyponatremia, hypercalcemia;
- i-hypersensitive to the components of the drug.
Isistim se-Hypothiazide
Isilinganisi sesilwanyana sikhethwe ngokuxhomekeka kwifom yesifo kunye nemeko yekhosi yayo. Iibhulile kufuneka zithathwe emva kokutya.
Kwiimeko ezininzi, ngokunyuka kwengcinezelo, ichiza lithathwa kwi-25-50 mg ngosuku. Umthamo weyeza lonyango lwe-symprome lingaba ngu-25-100 mg, kunye ne-Hypothiazide ithathwa kanye ngosuku okanye yonke imihla. Kwimeko ye-edema enzima, i-dose yokuqala yeziyobisi inganyuswa ibe yi-200 mg ngosuku. Kwi-premenstrual syndrome, njengomthetho, thabatha iipilisi eziyi-25 mg ngosuku.